Ator, Mark A: search on Z-Library

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1

The false vital sign: When pain levels are not predictive of discharge opioid prescriptions

Villwock, Jennifer A., Villwock, Mark R., New, Jacob, Ator, Gregory

Journal:

International Journal of Medical Informatics

Year:

2019

File:

PDF, 399 KB

2019

2

Long-Term Exposure to Oral Methylphenidate or dl-Amphetamine Mixture in Peri-Adolescent Rhesus Monkeys: Effects on Physiology, Behavior, and Dopamine System Development

Soto, Paul L, Wilcox, Kristin M, Zhou, Yun, Ator, Nancy A, Riddle, Mark A, Wong, Dean F, Weed, Michael R

Journal:

Neuropsychopharmacology

Year:

2012

Language:

english

File:

PDF, 817 KB

english, 2012

3

Characterizing cochlear mechano‐electric transduction using a nonlinear systems identification procedure

Chertoff, Mark E., Steele, Timothy, Ator, Gregory A., Bian, Lin

Journal:

The Journal of the Acoustical Society of America

Year:

1996

Language:

english

File:

PDF, 249 KB

english, 1996

4

Wake promoting agents: Search for next generation modafinil, lessons learned: Part III

Derek Dunn, Greg Hostetler, Mohamed Iqbal, Val R. Marcy, Yin Guo Lin, Bruce Jones, Lisa D. Aimone, John Gruner, Mark A. Ator, Edward R. Bacon, Sankar Chatterjee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 265 KB

english, 2012

5

Mechanism-based inactivation of horseradish peroxidase by sodium azide. Formation of meso-azidoprotoporphyrin IX

Ortiz de Montellano, Paul R., David, Shantha K., Ator, Mark A., Tew, David

Journal:

Year:

1988

Language:

english

File:

PDF, 874 KB

english, 1988

6

Wake-promoting agents: Search for next generation modafinil: Part I

Derek Dunn, Greg Hostetler, Mohamed Iqbal, Patricia Messina-McLaughlin, Alyssa Reiboldt, Yin Guo Lin, John Gruner, Edward R. Bacon, Mark A. Ator, Sankar Chatterjee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 219 KB

english, 2012

7

Wake-promoting agents: Search for next generation modafinil: Part II

Derek Dunn, Greg Hostetler, Mohamed Iqbal, Patricia Messina-McLaughlin, Alyssa Reiboldt, Yin Guo Lin, John Gruner, Edward R. Bacon, Mark A. Ator, Sankar Chatterjee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2012

Language:

english

File:

PDF, 186 KB

english, 2012

8

Design, Synthesis, and Biological Evaluation of Sulfonyl Acrylonitriles as Novel Inhibitors of Cancer Metastasis and Spread

Shen, Yi, Zificsak, Craig A., Shea, Jill E., Lao, Xuegang, Bollt, Oana, Li, Xiufen, Lisko, Joseph G., Theroff, Jay P., Scaife, Courtney L., Ator, Mark A., Ruggeri, Bruce A., Dorsey, Bruce D., Kuwada,

Journal:

Journal of Medicinal Chemistry

Year:

2015

Language:

english

File:

PDF, 928 KB

english, 2015

9

Combined inhibition of atypical PKC and histone deacetylase 1 is cooperative in basal cell carcinoma treatment

Mirza, Amar N., Fry, Micah A., Urman, Nicole M., Atwood, Scott X., Roffey, Jon, Ott, Gregory R., Chen, Bin, Lee, Alex, Brown, Alexander S., Aasi, Sumaira Z., Hollmig, Tyler, Ator, Mark A., Dorsey, Bru

Journal:

Year:

2017

Language:

english

File:

PDF, 1.54 MB

english, 2017

10

Preparation and evaluation of peptidic aspartyl hemiacetals as reversible inhibitors of interleukin-l β converting enzyme (ICE)

TODD L. GRAYBILL, ROLAND E. DOLLE, CARLA T. HELASZEK, ROBERT E. MILLER, MARK A. ATOR

Journal:

Chemical Biology & Drug Design

Year:

1994

Language:

english

File:

PDF, 948 KB

english, 1994

11

Mixed-Lineage Kinase 1 and Mixed-Lineage Kinase 3 Subtype-Selective Dihydronaphthyl[3,4-a]pyrrolo[3,4-c]carbazole-5-ones: Optimization, Mixed-Lineage Kinase 1 Crystallography, and Oral in Vivo Activity in 1-Methyl-4-phenyltetrahydropyridine Models

Hudkins, Robert L., Diebold, James L., Tao, Ming, Josef, Kurt A., Park, Chung Ho, Angeles, Thelma S., Aimone, Lisa D., Husten, Jean, Ator, Mark A., Meyer, Sheryl L., Holskin, Beverly P., Durkin, John

Journal:

Journal of Medicinal Chemistry

Year:

2008

Language:

english

File:

PDF, 751 KB

english, 2008

12

Corrigendum to “Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor” [Bioorg. Med. Chem. Lett. 21 (2011) 1991–1996]

Hamid R. Hoveyda, Marie-Odile Roy, Sebastien Blanc, Sophie Noël, Joseph M. Salvino, Mark A. Ator, Graeme Fraser

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 139 KB

english, 2011

13

2,7-Disubstituted-Pyrrolotriazine Kinase Inhibitors with an Unusually High Degree of Reactive Metabolite Formation

Wells-Knecht, Kevin J., Ott, Gregory R., Cheng, Mangeng, Wells, Gregory J., Breslin, Henry J., Gingrich, Diane E., Weinberg, Linda, Mesaros, Eugen F., Huang, Zeqi, Yazdanian, Mehran, Ator, Mark A., Ai

Journal:

Chemical Research in Toxicology

Year:

2011

Language:

english

File:

PDF, 1.55 MB

english, 2011

14

Synthesis, specificity, and antifungal activity of inhibitors of the Candida albicans .DELTA.24-sterol methyltransferase

Ator, Mark A., Schmidt, Stanley J., Adams, Jerry L., Dolle, Roland E., Kruse, Lawrence I., Frey, Carrie L., Barone, Janice M.

Journal:

Journal of Medicinal Chemistry

Year:

1992

Language:

english

File:

PDF, 1.01 MB

english, 1992

15

Aspartyl .alpha.-((1-Phenyl-3-(trifluoromethyl)- pyrazol-5-yl)oxy)methyl Ketones as Interleukin-1.beta. Converting Enzyme Inhibitors. Significance of the P1 and P3 Amido Nitrogens for Enzyme-Peptide Inhibitor Binding

Dolle, Roland E., Singh, Jasbir, Rinker, James, Hoyer, Denton, Prasad, C. V. C., Graybill, Todd L., Salvino, Joseph M., Helaszek, Carla T., Miller, Robert E., Ator, Mark A.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 464 KB

english, 1994

16

A highly selective, orally active inhibitor of Janus kinase 2, CEP-33779, ablates disease in two mouse models of rheumatoid arthritis

Kristine L Stump, Lily D Lu, Pawel Dobrzanski, Cynthia Serdikoff, Diane E Gingrich, Ben J Dugan, Thelma S Angeles, Mark S Albom, Mark A Ator, Bruce D Dorsey, Bruce A Ruggeri, Matthew M Seavey

Journal:

Arthritis Research & Therapy

Year:

2011

Language:

english

File:

PDF, 1.09 MB

english, 2011

17

Discovery and Characterization of 6-{4-[3-( R )-2-Methylpyrrolidin-1-yl)propoxy]phenyl}-2 H -pyridazin-3-one (CEP-26401, Irdabisant): A Potent, Selective Histamine H 3 Receptor Inverse Agonist

Hudkins, Robert L., Raddatz, Rita, Tao, Ming, Mathiasen, Joanne R., Aimone, Lisa D., Becknell, Nadine C., Prouty, Catherine P., Knutsen, Lars J. S., Yazdanian, Mehran, Moachon, Gilbert, Ator, Mark A.,

Journal:

Journal of Medicinal Chemistry

Year:

2011

Language:

english

File:

PDF, 1007 KB

english, 2011

18

Application of Genetic Algorithms to Combinatorial Synthesis: A Computational Approach to Lead Identification and Lead Optimization †,∇

Singh, Jasbir, Ator, Mark A., Jaeger, Edward P., Allen, Martin P., Whipple, David A., Soloweij, James E., Chowdhary, Swapan, Treasurywala, Adi M.

Journal:

Journal of the American Chemical Society

Year:

1996

Language:

english

File:

PDF, 450 KB

english, 1996

19

Pre-Steady-State and Steady-State Kinetic Analysis of E. coli Class I Ribonucleotide Reductase †

Ge, Jie, Yu, Guixue, Ator, Mark A., Stubbe, JoAnne

Journal:

Year:

2003

Language:

english

File:

PDF, 307 KB

english, 2003

20

First Examples of Peptidomimetic Inhibitors of Interleukin-1β Converting Enzyme

Dolle, Roland E., Prouty, Catherine P., Prasad, C. V. C., Cook, Ewell, Saha, Ashis, Ross, Tina Morgan, Salvino, Joseph M., Helaszek, Carla T., Ator, Mark A.

Journal:

Journal of Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 201 KB

english, 1996

21

Modification of CellSensor irf1- bla TF-1 and irf1- bla HEL Assays for Direct Comparison of Wild-Type JAK2 and JAK2 V617F Inhibition

Mason, Jennifer L., Holskin, Beverly P., Murray, Kristen A., Meyer, Sheryl L., Wells-Knecht, Kevin J., Ator, Mark A., Angeles, Thelma S.

Journal:

Assay and Drug Development Technologies

Year:

2011

Language:

english

File:

PDF, 469 KB

english, 2011

22

[The Enzymes] Volume 19 || 5 Mechanism-Based (Suicide) Enzyme Inactivation

Year:

1990

Language:

english

File:

PDF, 3.27 MB

english, 1990

23

Comparative Study of Transport Processes of Nitrogen, Phosphorus, and Herbicides to Streams in Five Agricultural Basins, USA

Domagalski, Joseph L., Ator, Scott, Coupe, Richard, McCarthy, Kathleen, Lampe, David, Sandstrom, Mark, Baker, Nancy

Journal:

Journal of Environmental Quality

Year:

2008

Language:

english

File:

PDF, 921 KB

english, 2008

24

Calpain inhibitors based on the quiescent affinity label concept: high rates of calpain inactivation with leaving groups derived from N-hydroxy peptide coupling reagents

Rabindranath Tripathy, Mark A. Ator, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2000

Language:

english

File:

PDF, 143 KB

english, 2000

25

P1 Aspartate-Based Peptide .alpha.-((2,6-Dichlorobenzoyl)oxy)methyl Ketones as Potent Time-Dependent Inhibitors of Interleukin-1.beta.-Converting Enzyme

Dolle, Roland E., Hoyer, Denton, Prasad, C. V. C., Schmidt, Stanley J., Helaszek, Carla T., Miller, Robert E., Ator, Mark A.

Journal:

Journal of Medicinal Chemistry

Year:

1994

Language:

english

File:

PDF, 291 KB

english, 1994

26

Lead development: Validation and application of high throughput screening for determination of pharmacokinetic parameters for enzyme inhibitors

Jasbir Singh, Jim Soloweij, Martin Allen, Loran Killar, Mark Ator

Journal:

Bioorganic & Medicinal Chemistry

Year:

1996

Language:

english

File:

PDF, 430 KB

english, 1996

27

A New Class of Potent Vascular Endothelial Growth Factor Receptor Tyrosine Kinase Inhibitors: Structure−Activity Relationships for a Series of 9-Alkoxymethyl-12-(3-hydroxypropyl)indeno[2,1- a ]pyrrolo[3,4- c ]carbazole-5-ones and the Identification of CEP-5214 and Its Dimethylglycine Ester Prodrug Clinical Candidate CEP-7055

Gingrich, Diane E., Reddy, Dandu R., Iqbal, Mohamed A., Singh, Jasbir, Aimone, Lisa D., Angeles, Thelma S., Albom, Mark, Yang, Shi, Ator, Mark A., Meyer, Sheryl L., Robinson, Candy, Ruggeri, Bruce A.,

Journal:

Journal of Medicinal Chemistry

Year:

2003

Language:

english

File:

PDF, 414 KB

english, 2003

28

The false vital sign: When pain levels are not predictive of discharge opioid prescriptions

Villwock, Jennifer A., Villwock, Mark R., New, Jacob, Ator, Gregory

Journal:

International Journal of Medical Informatics

Year:

2019

Language:

english

File:

PDF, 399 KB

english, 2019

29

Aequorin functional assay for characterization of G-protein-coupled receptors: Implementation with cryopreserved transiently transfected cells

Bruce Jones, Beverly Holskin, Sheryl Meyer, Thao Ung, Vincent Dupriez, Sandra Y. Flores, Emmanuel Burgeon, Mark Ator, Emir Duzic

Journal:

Analytical Biochemistry

Year:

2010

Language:

english

File:

PDF, 462 KB

english, 2010

30

Discovery of 3-aryl-5-acylpiperazinyl-pyrazoles as antagonists to the NK3 receptor

Hamid R. Hoveyda, Marie-Odile Roy, Sebastien Blanc, Sophie Noël, Joseph M. Salvino, Mark A. Ator, Graeme Fraser

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2011

Language:

english

File:

PDF, 609 KB

english, 2011

31

3-chloro-4-carboxamido-6-arylpyridazines as a non-peptide class of interleukin-1β converting enzyme inhibitor

Roland E. Dolle, Denton Hoyer, James M. Rinker, Tina Morgan Ross, Stanley J. Schmidt, Carla T. Helaszek, Mark A. Ator

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1997

Language:

english

File:

PDF, 182 KB

english, 1997

32

Synthesis and Biological Activity of a Series of Potent Fluoromethyl Ketone Inhibitors of Recombinant Human Calpain I

Chatterjee, Sankar, Ator, Mark A., Bozyczko-Coyne, Donna, Josef, Kurt, Wells, Gregory, Tripathy, Rabindranath, Iqbal, Mohamed, Bihovsky, Ron, Senadhi, Shobha E., Mallya, Satish, O'Kane, Teresa M., McK

Journal:

Journal of Medicinal Chemistry

Year:

1997

Language:

english

File:

PDF, 240 KB

english, 1997

33

P′-extended α-ketoamide inhibitors of proteasome

Sankar Chatterjee, Derek Dunn, Satish Mallya, Mark A. Ator

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 184 KB

english, 1999

34

Mixed lineage kinase activity of indolocarbazole analogues

Chikara Murakata, Masami Kaneko, George Gessner, Thelma S Angeles, Mark A Ator, Teresa M O'Kane, Beth Ann W McKenna, Beth Ann Thomas, Joanne R Mathiasen, Michael S Saporito, Donna Bozyczko-Coyne, Robe

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

2002

Language:

english

File:

PDF, 164 KB

english, 2002

35

From an Atypical Wake-promoting Agent to Potent Histamine-3 Receptor Inverse Agonists

Dunn, Derek, Raddatz, Rita, Ator, Mark A., Bacon, Edward R., Chatterjee, Sankar

Journal:

Chemical Biology & Drug Design

Year:

2013

Language:

english

File:

PDF, 328 KB

english, 2013

36

Comparison of Two Homogeneous Cell-Based Kinase Assays for JAK2 V617F: SureFire pSTAT5 and GeneBLAzer Fluorescence Resonance Energy Transfer Assays

Qian, Jie, Mason, Jennifer L., Holskin, Beverly P., Murray, Kristen A., Meyer, Sheryl L., Ator, Mark A., Angeles, Thelma S.

Journal:

Assay and Drug Development Technologies

Year:

2012

Language:

english

File:

PDF, 309 KB

english, 2012

37

P2-achiral, P'-extended α-ketoamide inhibitors of calpain I

Sankar Chatterjee, Derek Dunn, Ming Tao, Gregory Wells, Zi-Qiang Gu, Ron Bihovsky, Mark A. Ator, Robert Siman, John P. Mallamo

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1999

Language:

english

File:

PDF, 209 KB

english, 1999

38

Laquinimod arrests experimental autoimmune encephalomyelitis by activating the aryl hydrocarbon receptor

Kaye, Joel, Piryatinsky, Victor, Birnberg, Tal, Hingaly, Tal, Raymond, Emanuel, Kashi, Rina, Amit-Romach, Einat, Caballero, Ignacio S., Towfic, Fadi, Ator, Mark A., Rubinstein, Efrat, Laifenfeld, Daph

Journal:

Proceedings of the National Academy of Sciences

Year:

2016

Language:

english

File:

PDF, 1.41 MB

english, 2016

39

Synthesis and evaluation of diacylhydrazines as inhibitors of the interleukin-1β converting enzyme (ICE)

Todd L. Graybill, Roland E. Dolle, Carla T. Helaszek, Mark A. Ator, Joost Strasters

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1995

Language:

english

File:

PDF, 374 KB

english, 1995

40

Comparison of LanthaScreen Eu Kinase Binding Assay and Surface Plasmon Resonance Method in Elucidating the Binding Kinetics of Focal Adhesion Kinase Inhibitors

Mason, Jennifer L., Spais, Chrysanthe, Husten, Jean, Prouty, Eric, Albom, Mark S., Meyer, Sheryl L., Ator, Mark A., Angeles, Thelma S.

Journal:

Assay and Drug Development Technologies

Year:

2012

Language:

english

File:

PDF, 310 KB

english, 2012

41

A Sensitive, Continuously Recording Fluorogenic Assay for Calpain

Satish K. Mallya, Sheryl Meyer, Donna Bozyczko–Coyne, Robert Siman, Mark A. Ator

Journal:

Biochemical and Biophysical Research Communications

Year:

1998

Language:

english

File:

PDF, 76 KB

english, 1998

42

σRecognition sites in brain and peripheral tissues Characterization and effects of cytochrome P450 inhibitors

Diane L. DeHaven-Hudkins, Lorraine F. Lanyon, Felicia Y. Ford-Rice, Mark A. Ator

Journal:

Biochemical Pharmacology

Year:

1994

Language:

english

File:

PDF, 862 KB

english, 1994

43

Mechanism of inactivation of Escherichia coli ribonucleotide reductase by 2'-chloro-2'-deoxyuridine 5'-diphosphate: evidence for generation of a 2'-deoxy-3'-ketonucleotide via a net 1,2 hydrogen shift

Ator, Mark A., Stubbe, JoAnne

Journal:

Year:

1985

Language:

english

File:

PDF, 1.64 MB

english, 1985

44

ChemInform Abstract: Calpain Inhibitors Based on the Quiescent Affinity Label Concept: High Rates of Calpain Inactivation with Leaving Groups Derived from N-Hydroxy Peptide Coupling Reagents.

Rabindranath Tripathy, Mark A. Ator, John P. Mallamo

Journal:

Year:

2001

File:

PDF, 30 KB

2001

45

Potent fluoromethyl ketone inhibitors of recombinant human calpain I

Sankar Chatterjee, Kurt Josef, Gregory Wells, Mohamed Iqbal, Ron Bihovsky, John P. Mallamo, Mark A. Ator, Donna Bozyczko-Coyne, Satish Mallya, Shobha Senadhi, Robert Siman

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1996

Language:

english

File:

PDF, 230 KB

english, 1996

46

P2-proline-derived inhibitors of calpain I

Rabindranath Tripathy, Zi-Qiang Gu, Derek Dunn, Shobha E. Senadhi, Mark A. Ator, Sankar Chatterjee

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1998

Language:

english

File:

PDF, 235 KB

english, 1998

47

Synthesis and evaluation of azapeptide-derived inhibitors of serine and cysteine proteases

Todd L. Graybill, Mitchell J. Ross, Bruce R. Gauvin, Jill S. Gregory, Alex L. Harris, Mark A. Ator, James M. Rinker, Roland E. Dolle

Journal:

Bioorganic & Medicinal Chemistry Letters

Year:

1992

Language:

english

File:

PDF, 473 KB

english, 1992

48

Indices of endolymphatic hydrops derived from measures of cochlear mechanics

Gregory A. Ator, Lin Bian, Mark E. Chertoff

Journal:

Otolaryngology - Head and Neck Surgery

Year:

1996

Language:

english

File:

PDF, 108 KB

english, 1996

49

Serendipitous Discovery of a Prodrug of a PARP-1 Inhibitor

Dunn, Derek, Husten, Jean, Aimone, Lisa D., Ator, Mark A., Chatterjee, Sankar

Journal:

Chemical Biology & Drug Design

Year:

2013

Language:

english

File:

PDF, 97 KB

english, 2013

50

d -Amino Acid Containing, High-Affinity Inhibitors of Recombinant Human Calpain I †

Chatterjee, Sankar, Gu, Zi-Qiang, Dunn, Derek, Tao, Ming, Josef, Kurt, Tripathy, Rabindranath, Bihovsky, Ron, Senadhi, Shobha E., O'Kane, Teresa M., McKenna, Beth Ann, Mallya, Satish, Ator, Mark A., B

Journal:

Journal of Medicinal Chemistry

Year:

1998

Language:

english

File:

PDF, 56 KB

english, 1998

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